In vitro cytotoxicity studies of palladacyclic complexes containing the

The reactions between [Pd2{(C,N)eC6H4CH2NH(Et)}2(m-X)2] (X ¼ Cl or Br) and 1,2-

bis(diphenylphosphino)ethane (dppe) in the 1:1 molar ratio resulted in the dppe-bridged Pd(II) complexes,

[Pd2{(C,N)eC6H4CH2NH(Et)}2(m-dppe)(Cl)2] (1) and [Pd2{(C,N)eC6H4CH2NH(Et)}2(m-dppe)(Br)2]

(2), respectively, which were characterized by elemental analyses, infrared (IR), 1H- and 31P{1H} NMR

spectroscopy. The molecular structure of 1 was determined by single-crystal X-ray diffraction. In vitro

cytotoxicity of 1, 2, dppe, PhCH2NH(Et) and cisplatin were carried out against four human tumor cell

lines. The interactions of complexes towards DNA and protein are investigated. The results suggested that

both complexes could interact with FS-DNA through the intercalation mode. Moreover, the reactivity

towards BSA revealed that the microenvironment and the secondary structure of BSA were changed in

the presence of Pd(II) complexes.

https://people.iut.ac.ir/en/karami/content/vitro-cytotoxicity-studies-palladacyclic-complexes-containing